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{ "complex_dir": "1433B_HUMAN_1_240_pep_0", "ligand_original_name": "2bq0_A_rec_5f74_amp_lig_it1_it2_tt_docked.sdf.gz", "pair_idx": 0, "receptor_path": "1433B_HUMAN_1_240_pep_0/2bq0_A_rec.pdb", "source_type": "cdonly" }
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hf://datasets/kohbanye/crossdocked2020@8361e55b96939a57b7ad27e04b3b5bcb09f87f93/ligands/000000.tar
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hf://datasets/kohbanye/crossdocked2020@8361e55b96939a57b7ad27e04b3b5bcb09f87f93/ligands/000000.tar
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CrossDocked2020

Pre-processed CrossDocked2020 dataset containing raw receptor PDB and ligand SDF.gz files, organized for efficient loading.

Dataset Summary

  • Unique pairs: 25,092,018
  • Unique receptor PDB files: 24,533
  • Source types: cdonly, it0, it2_redocked
  • Fold splits: 3 folds (0, 1, 2) per source type category

Repository Structure

receptors/          Unique receptor PDB files in tar.gz archives
ligands/            Ligand SDF.gz files in tar shards (WebDataset-compatible)
manifest.parquet    Pair index with metadata and fold split info

Ligand Tar Shard Format

Each shard is a tar file containing pairs of files per sample:

  • {pair_idx:07d}.sdf.gz — original ligand SDF.gz (all conformers)
  • {pair_idx:07d}.json — metadata (receptor_path, complex_dir, source_type)

Manifest Schema

Column Type Description
pair_idx uint32 Global unique pair ID
complex_dir string Complex directory name
receptor_pdb string Receptor PDB filename
ligand_sdf_gz string Ligand SDF.gz filename
source_type string cdonly / it0 / it2_redocked
shard_idx uint16 Ligand shard number
label int8 Types file label (0/1)
score1 float32 Types file score 1
score2 float32 Types file score 2
{cat}_fold{n} string "train" / "test" per category and fold

Original Source

Paul G. Francoeur, Tomohide Masuda, Jocelyn Sunseri, Andrew Jia, Richard B. Iovanisci, Ian Snyder, David R. Koes. J. Chem. Inf. Model. 2020, 60(9), p.4200–4215.

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